SCHEMBL8113999

SCHEMBL8113999

CCOC(=O)CC1COC(c2ccccc2Cl)c2cc(Cl)ccc2N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
POLB P06746 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP3A4 P08684 2/20 0.38
ALOX12 P18054 1/20 0.38
RAB9A P51151 3/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPK1 P28482 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ATM Q13315 1/20 0.37
MAPT P10636 3/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111295 0.76 ALDH1A1 (0.43) TSHRPOLBCYP2C9CYP2C19CYP3A4
SCHEMBL8116509 0.76 ALDH1A1 (0.41) TSHRPOLBRAB9AALDH1A1SMN1; SMN2
SCHEMBL6766521 0.70 TSHR (0.46) TSHRPOLBCYP1A2CYP2C9CYP2C19
SCHEMBL8116269 0.70 MAPT (0.50) TSHRPOLBCYP1A2CYP2C9CYP2C19
SCHEMBL6949285 0.69 TSHR (0.44) TSHRPOLBCYP1A2CYP2C9CYP2C19
SCHEMBL7302983 0.68 L3MBTL1 (0.47) TSHRPOLBCYP1A2ALDH1A1SMN1; SMN2
SCHEMBL6952331 0.68 ALDH1A1 (0.47) TSHRALDH1A1SMN1; SMN2MAPTHTT
SCHEMBL6952325 0.68 ALDH1A1 (0.47) TSHRALDH1A1SMN1; SMN2MAPTHTT
SCHEMBL4124441 0.67 CDYL2 (0.44) RAB9AMEN1KMT2AATMFDFT1
SCHEMBL4123224 0.67 FDFT1 (0.39) ALDH1A1MAPK1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645378-B1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-08-23 EP claimed
EP-0645378-B1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-08-23 EP disclosed
US-5698691-A ANTICHOLESTEROL AGENT; SYNTHETASE INHIBITOR; FUNGICIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-16 US disclosed
EP-0645378-A1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors Takeda Chemical Industries, Ltd. (JP) 1995-03-29 EP disclosed