SCHEMBL8123714

SCHEMBL8123714

O=C1CCCCN1C1=CC(CF)(CF)Oc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
POLB P06746 1/20 0.37
APEX1 P27695 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
GAA P10253 1/20 0.35
CASP3 P42574 3/20 0.34
CASP1 P29466 2/20 0.34
CASP4 P49662 2/20 0.34
CASP7 P55210 2/20 0.34
CASP9 P55211 2/20 0.34
RAB9A P51151 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
CAPN9 O14815 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
CASP8 Q14790 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8120777 0.97 CASP6 (0.37) CASP6TDP1POLBAPEX1CTDSP1
SCHEMBL10757454 0.82 CASP6 (0.40) CASP6TDP1POLBAPEX1CTDSP1
SCHEMBL8130025 0.81 LIPE (0.34) KMT2AALDH1A1MEN1GAAHRH3
SCHEMBL8862309 0.80 PDK2 (0.31)
SCHEMBL8130641 0.80 PDE4A (0.38) ALDH1A1CASP3MALT1HRH3
SCHEMBL8130743 0.80 PDK2 (0.30)
SCHEMBL8862306 0.80 PDK2 (0.30)
SCHEMBL9735458 0.78 NR1H4 (0.39) CASP6TDP1POLBAPEX1CTDSP1
SCHEMBL8130800 0.78
SCHEMBL8131501 0.78 PDK2 (0.34) KMT2AALDH1A1MEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655448-B1 BENZOPYRAN AND BENZOXAZINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2000-04-12 EP disclosed
US-5977167-A Benzopyran and benzoxazine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1999-11-02 US disclosed
US-5874446-A ANTIASTHMATICS, ANTIEPILEPSY AGENTS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1999-02-23 US disclosed
US-5614633-A POTASSIUM CHANNEL ACTIVATOR CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1997-03-25 US disclosed
EP-0655448-A1 BENZOPYRAN AND BENZOXAZINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-05-31 EP disclosed