SCHEMBL8130641

SCHEMBL8130641

N#Cc1ccc2c(c1)C(N1CCCCC1=O)=CC(CF)(CF)O2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
ABCC9 O60706 2/20 0.38
ABCC8 Q09428 2/20 0.38
KCNJ11 Q14654 2/20 0.38
KCNJ8 Q15842 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.38
HTR2A P28223 1/20 0.36
HTR1A P08908 2/20 0.35
CHEK1 O14757 1/20 0.33
F10 P00742 1/20 0.33
CASP3 P42574 1/20 0.33
PTGER4 P35408 1/20 0.32
MALT1 Q9UDY8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8130466 0.97 ABCC9 (0.41) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL10759518 0.84 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8130025 0.82 LIPE (0.34) KDM4EALDH1A1HRH3
SCHEMBL8862309 0.81 PDK2 (0.31)
SCHEMBL9139375 0.81 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8862306 0.80 PDK2 (0.30)
SCHEMBL8130743 0.80 PDK2 (0.30)
SCHEMBL8123714 0.80 CASP6 (0.37) CASP3MALT1ALDH1A1HRH3
SCHEMBL8130800 0.79
SCHEMBL8131501 0.79 PDK2 (0.34) LMNAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655448-B1 BENZOPYRAN AND BENZOXAZINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2000-04-12 EP disclosed
US-5977167-A Benzopyran and benzoxazine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1999-11-02 US disclosed
US-5874446-A ANTIASTHMATICS, ANTIEPILEPSY AGENTS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1999-02-23 US disclosed
US-5614633-A POTASSIUM CHANNEL ACTIVATOR CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1997-03-25 US disclosed
EP-0655448-A1 BENZOPYRAN AND BENZOXAZINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-05-31 EP disclosed