SCHEMBL8124407

SCHEMBL8124407

O=C(c1cccc([N+](=O)[O-])c1)c1c(Cl)cccc1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
TSHR P16473 2/20 0.58
CES2 O00748 1/20 0.57
CES1 P23141 1/20 0.57
TP53 P04637 1/20 0.55
VCAM1 P19320 2/20 0.51
MAPT P10636 1/20 0.51
MAPK1 P28482 1/20 0.51
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
CRHBP P24387 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27511511 0.84 VCAM1 (0.60) ALDH1A1TSHRVCAM1MAPTMAPK1
SCHEMBL8622869 0.82 VCAM1 (0.77) ALDH1A1TSHRCES2CES1TP53
SCHEMBL10903202 0.81 ALDH1A1 (0.56) ALDH1A1TSHRCES2CES1TP53
SCHEMBL4254988 0.81 NPC1 (0.63) ALDH1A1TSHRCES2CES1TP53
SCHEMBL30192262 0.81 NPC1 (0.63) ALDH1A1TSHRCES2CES1TP53
SCHEMBL181572 0.81 CES2 (0.78) ALDH1A1TSHRCES2CES1TP53
SCHEMBL8962468 0.79 CES2 (0.75) ALDH1A1TSHRCES2CES1TP53
SCHEMBL10341585 0.79 CES2 (0.60) ALDH1A1TSHRCES2CES1TP53
SCHEMBL14984180 0.78 ALDH1A1 (0.68) ALDH1A1TSHRCES2CES1TP53
SCHEMBL10902888 0.78 TSHR (0.59) ALDH1A1TSHRCES2CES1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973777-A1 FUROPYRIDINE, THIENOPYRIDINE, PYRROLOPYRIDINE AND RELATED PYRIMIDINE, PYRIDAZINE AND TRIAZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-01-26 EP disclosed
US-6001849-A Furopyridine, thienopyridine pyrrolopyridine useful in controlling chemical synaptic transmission ABBOTT LABORATORIES (US) 1999-12-14 US disclosed
EP-0934308-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 1999-08-11 EP disclosed
WO-1998046609-A1 FUROPYRIDINE, THIENOPYRIDINE, PYRROLOPYRIDINE AND RELATED PYRIMIDINE, PYRIDAZINE AND TRIAZINE COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1998-10-22 WO disclosed
WO-1997046554-A1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1997-12-11 WO disclosed