SCHEMBL8127484

SCHEMBL8127484

c1ccc(CNc2ncc3ncncc3n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.50
ATM Q13315 1/20 0.47
RAD52 P43351 1/20 0.46
ALDH1A1 P00352 5/20 0.46
CYP1A2 P05177 5/20 0.46
CYP3A4 P08684 5/20 0.46
CYP2D6 P10635 5/20 0.46
ALOX15 P16050 4/20 0.46
CYP2C19 P33261 4/20 0.46
TSHR P16473 4/20 0.46
LMNA P02545 2/20 0.45
GALR3 O60755 2/20 0.45
NR2F2 P24468 2/20 0.45
KMT2A Q03164 2/20 0.45
APP P05067 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
PKM P14618 1/20 0.45
UBE2N P61088 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7951301 0.81 VNN1 (0.50) EGFRNR2F2KMT2AAPPMAPT
SCHEMBL27857007 0.77 RAD52 (0.56) ATMRAD52ALDH1A1LMNAKMT2A
SCHEMBL9116416 0.75 EGFR (0.54) EGFRATMRAD52ALDH1A1CYP1A2
SCHEMBL9779691 0.74 FABP1 (0.52) EGFRALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5934943 0.73 RAB9A (0.57) EGFRALDH1A1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL28584936 0.72 KCNH3 (0.52) EGFRALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL1019383 0.72 IP6K1 (0.47) ATMRAD52ALDH1A1CYP1A2CYP2D6
SCHEMBL8674551 0.72 CDK1 (0.59) ALDH1A1CYP1A2CYP3A4CYP2D6ALOX15
SCHEMBL29893789 0.71 RAB9A (0.48) ATMRAD52ALDH1A1LMNAKMT2A
SCHEMBL6837276 0.71 EGFR (0.57) EGFRATMRAD52ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971925-A1 PYRIMIDOPYRIMIDINE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 2000-01-19 EP disclosed
WO-1998043974-A1 PYRIMIDOPYRIMIDINE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1998-10-08 WO disclosed