SCHEMBL8128162

SCHEMBL8128162

COCCOCOc1c(F)ccc(OC(=O)COc2cccc3c2C(=O)NC3=O)c1OCOCCOC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
RARG P13631 1/20 0.33
PTPN1 P18031 1/20 0.32
GAA P10253 4/20 0.32
MAPT P10636 4/20 0.32
FFAR4 Q5NUL3 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KCNN4 O15554 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8119171 0.91 CASP3 (0.36) CASP3DDB1CRBNRARGPTPN1
SCHEMBL8132547 0.86 CYP1A2 (0.34) CASP3DDB1CRBNRARGGAA
SCHEMBL8167098 0.86 GAA (0.34) CASP3DDB1CRBNRARGGAA
SCHEMBL8134794 0.81 RARG (0.35) CASP3DDB1CRBNRARGGAA
SCHEMBL7963652 0.80 CASP3 (0.33) CASP3RARGGAAFFAR4ALDH1A1
SCHEMBL9416166 0.79 CASP3 (0.31) CASP3DDB1CRBN
SCHEMBL8132902 0.78 AR (0.34) CASP3DDB1CRBNGAAALDH1A1
SCHEMBL7959787 0.74 PTGS1 (0.36) CASP3RARGGAAFFAR4ALDH1A1
SCHEMBL8133598 0.74 PTPN1 (0.47) RARGPTPN1GAAALDH1A1HPGD
SCHEMBL7967343 0.73 FABP4 (0.38) CASP3RARGGAAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0551034-B1 Antibiotic cephalosporins having in position 7 a substituted benzyloxyimino radical HOECHST MARION ROUSSEL INC (FR) 2000-09-20 EP disclosed
EP-1016646-A1 Intermediates for the preparation of cephalosporines containing on the 7-position a substituted benzyloximino radical HOECHST MARION ROUSSEL (FR) 2000-07-05 EP disclosed
EP-0551034-A2 Cephalosporins having in position 7 a benzyloxyimino radical substitute, process for their preparation and their use as medicaments ROUSSEL UCLAF (FR) 1993-07-14 EP disclosed