SCHEMBL8129109

SCHEMBL8129109

O=[N+]([O-])C=C(NCc1cccc(Cl)c1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
MAPT P10636 3/20 0.47
HTT P42858 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
MYC P01106 1/20 0.45
MAX P61244 1/20 0.45
EPHX2 P34913 1/20 0.43
P2RX1 P51575 5/20 0.43
LMNA P02545 2/20 0.43
HPGD P15428 1/20 0.43
ATG4B Q9Y4P1 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
PLA2G1B P04054 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
P2RX4 Q99571 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8129106 1.00 MEN1 (0.47) MEN1KMT2AMAPTHTTNPSR1
SCHEMBL8129009 0.87 ATG4B (0.45) MEN1KMT2AMAPTLMNAHPGD
SCHEMBL8129006 0.87 ATG4B (0.45) MEN1KMT2AMAPTLMNAHPGD
SCHEMBL8134160 0.82 TP53 (0.47) MEN1KMT2AMAPTHTTNPSR1
SCHEMBL8134161 0.82 TP53 (0.47) MEN1KMT2AMAPTHTTNPSR1
SCHEMBL3305997 0.77 MYC (0.74) MEN1KMT2AMAPTHTTNPSR1
SCHEMBL8129144 0.72 P2RX1 (0.39) MEN1KMT2AMAPTP2RX1LMNA
SCHEMBL8129143 0.72 P2RX1 (0.39) MEN1KMT2AMAPTP2RX1LMNA
SCHEMBL8138760 0.72 ALDH1A1 (0.41) MEN1KMT2AMAPTHTTP2RX1
SCHEMBL8138758 0.72 ALDH1A1 (0.41) MEN1KMT2AMAPTHTTP2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147098-A USEFUL IN THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM, CARDIOVASCULAR SYSTEM, PULMONARY SYSTEM, GASTROINTESTINAL SYSTEM AND ENDOCRINOLOGIC SYSTEM NOVO NORDISK A/S (DK) 2000-11-14 US disclosed