SCHEMBL8133530

SCHEMBL8133530

CN1CCc2c(-c3ccc(S(N)(=O)=O)cc3)cc3c(c2C1)NC(=O)C3=O

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.40
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
CA12 O43570 2/20 0.39
PTGS1 P23219 1/20 0.37
GRIA1 P42261 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIA3 P42263 1/20 0.37
GRIA4 P48058 1/20 0.37
HTR6 P50406 4/20 0.34
CA4 P22748 1/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8126477 0.89 GRIA1 (0.38) PTGS2CA1CA2CA9CA12
SCHEMBL8126480 0.89 GRIA1 (0.38) PTGS2CA1CA2CA9CA12
SCHEMBL4370479 0.88 HTR6 (0.47) GRIA1GRIA2GRIA3GRIA4HTR6
SCHEMBL6609340 0.86 CASP3 (0.47) HTR6BRD4
SCHEMBL8134987 0.85 SMN1; SMN2 (0.42) GRIA1GRIA2GRIA3GRIA4HTR6
SCHEMBL13592440 0.85 GRIA1 (0.36) GRIA1GRIA2GRIA3GRIA4
SCHEMBL8102934 0.85 CES1 (0.39) GRIA1GRIA2GRIA3GRIA4HTR6
SCHEMBL6609831 0.85 MCHR1 (0.39) GRIA1GRIA2GRIA3GRIA4
SCHEMBL6607897 0.85 CYP2C9 (0.39) GRIA1GRIA2GRIA3GRIA4HTR6
SCHEMBL8136178 0.84 MEN1 (0.36) GRIA1GRIA2GRIA3GRIA4HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781285-B1 FUSED INDOLE AND QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE AS GLUTAMATE ANTAGONISTS NEUROSEARCH AS (DK) 2000-01-12 EP disclosed
US-5801174-A CEREBROVASCULAR DISORDERS NEUROSEARCH A/S (DK) 1998-09-01 US disclosed
WO-1996008495-A1 FUSED INDOLE AND QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1996-03-21 WO disclosed