SCHEMBL8134166

SCHEMBL8134166

COc1[c]ccc(S(=O)(=O)C(C)C)c1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 1/20 0.32
POLB P06746 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL358028 0.80 SMN1; SMN2 (0.46) POLBTSHRMAPK1
SCHEMBL8129522 0.79 MMP13 (0.38)
SCHEMBL7045277 0.79 ALDH1A1 (0.36) POLBTSHRMAPK1
SCHEMBL26688580 0.77 PSIP1 (0.39)
SCHEMBL17291118 0.77 ABL1 (0.31)
SCHEMBL3305889 0.76 MAPT (0.49) POLBTSHRMAPK1
SCHEMBL16880017 0.75 HRH4 (0.33) POLB
SCHEMBL7476629 0.75 ALDH1A1 (0.42) POLB
SCHEMBL29287789 0.74 LOX (0.35)
SCHEMBL28247559 0.72 ALDH1A1 (0.54) POLBTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0763524-B1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO CO (JP) 2000-08-23 EP disclosed
US-6040339-A TREATMENT AND PROPHYLAXIS OF HYPERCHOLESTEREMIA OR ARTERIOSCLEROSIS IN A MAMMAL SANKYO COMPANY, LIMITED (JP) 2000-03-21 US disclosed
US-5880147-A Amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prohylactic use SANKYO COMPANY, LIMITED (JP) 1999-03-09 US disclosed
EP-0763524-A1 Urea and amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use SANKYO COMPANY LIMITED (JP) 1997-03-19 EP disclosed