Cyclooctane

Cyclooctane

SCHEMBL8134205

C1CCCCCCC1.Fc1ccc(Nc2ccc(F)cc2)cc1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.45
TDP1 Q9NUW8 3/20 0.45
FKBP1A P62942 1/20 0.45
GLA P06280 1/20 0.45
KCNH3 Q9ULD8 1/20 0.45
GRM5 P41594 1/20 0.44
GRM1 Q13255 1/20 0.44
MEN1 O00255 3/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
MAPK10 P53779 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
ALOX12 P18054 1/20 0.43
PTGS1 P23219 1/20 0.43
SLC6A2 P23975 1/20 0.43
MAPK1 P28482 1/20 0.43
PTGS2 P35354 1/20 0.43
HTR2B P41595 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL395770 0.91 ALDH1A1 (0.50) KMT2ATDP1KCNH3MEN1POLB
SCHEMBL21560850 0.82 TXN (0.57) KMT2ATDP1KCNH3MEN1POLB
SCHEMBL4579384 0.82 TXN (0.57) KMT2ATDP1KCNH3MEN1POLB
SCHEMBL904596 0.80 ALDH1A1 (0.72) KMT2ATDP1KCNH3MEN1POLB
SCHEMBL25354895 0.78 MEN1 (0.59) KMT2ATDP1MEN1POLBALDH1A1
SCHEMBL25500981 0.78 MAPT (0.61) KMT2ATDP1MEN1POLBALDH1A1
SCHEMBL14463321 0.78 ACHE (0.68) KMT2ATDP1KCNH3MEN1MAPT
SCHEMBL20036881 0.78 MEN1 (0.41) KMT2ATDP1KCNH3MEN1POLB
SCHEMBL1028204 0.78 GAA (0.61) KMT2ATDP1MEN1POLBALDH1A1
SCHEMBL10569084 0.76 MEN1 (0.61) KMT2ATDP1KCNH3MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042291-A1 ARYL-SUBSTITUTED PYRIDYLALKANE, ALKENE, AND ALKINE CARBOXAMIDES USEFUL AS CYTOSTATIC AND IMMUNOSUPPRESSIVE AGENTS Klinge Pharma GmbH (DE) 2000-10-11 EP disclosed
WO-1999031064-A1 ARYL-SUBSTITUTED PYRIDYLALKANE, ALKENE, AND ALKINE CARBOXAMIDES USEFUL AS CYTOSTATIC AND IMMUNOSUPPRESSIVE AGENTS KLINGE PHARMA GMBH (DE) 1999-06-24 WO disclosed