SCHEMBL8136108

SCHEMBL8136108

Cc1cc(CCCOc2ccc(C(=N)NO)cc2C(F)(F)F)on1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
S1PR1 P21453 18/20 0.42
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875008 0.86 NR1I2 (0.41) NR1I2CYP3A4CYP2D6THRATHRB
SCHEMBL8136112 0.82 NR1I2 (0.45) NR1I2CYP3A4CYP2D6S1PR1THRA
SCHEMBL8876220 0.80 HDAC6 (0.46) NR1I2CYP3A4CYP2D6
SCHEMBL8136126 0.80 PRSS1 (0.49) THRATHRB
SCHEMBL23588051 0.79 THRA (0.52) S1PR1THRATHRB
SCHEMBL19411800 0.77 THRA (0.58) S1PR1THRATHRB
SCHEMBL13139482 0.77 THRA (0.58) S1PR1THRATHRB
SCHEMBL8136926 0.77 NR1I2 (0.45) NR1I2CYP3A4CYP2D6S1PR1
SCHEMBL10507968 0.76 NR1I2 (0.44) NR1I2CYP3A4CYP2D6S1PR1THRA
SCHEMBL8875413 0.76 NR1I2 (0.47) NR1I2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0566199-B1 1,2,4-Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents SANOFI SA (FR) 2000-03-01 EP disclosed
US-5643929-A TREATMENT OF PICORNAVIRAL OR RHINOVIRUS AND CHEMICAL INTERMEDIATES SANOFI WINTHROP, INC. (US) 1997-07-01 US disclosed
US-5464848-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1995-11-07 US disclosed
US-5349068-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1994-09-20 US disclosed
EP-0566199-A1 1,2,4-Oxadiazolyl-phenoxyalkylisoxazoles and their use a s antiviral agents STERLING WINTHROP INC. (US) 1993-10-20 EP disclosed