SCHEMBL8140405

SCHEMBL8140405

CN1CC=C(c2csc3ccc(N(C(N)=O)c4ccc(-c5ccncc5)c5ccccc45)cc23)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.35
HTR1A P08908 2/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
NOS3 P29474 3/20 0.33
NOS1 P29475 3/20 0.33
NOS2 P35228 3/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
ALOX15 P16050 1/20 0.33
SLC6A4 P31645 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994311 0.76 ERN1 (0.43) HTR6HTR1AHTR1DHTR1BNOS3
SCHEMBL6994397 0.72 BLM (0.39) NOS3NOS1KDM4ELMNAPOLB
SCHEMBL7718815 0.70 HTR1D (0.46) HTR6HTR1AHTR1DHTR1BNOS3
SCHEMBL11874262 0.70 HTR6 (0.55) HTR6HTR1AKDM4ELMNAPOLB
SCHEMBL8658544 0.68 NOS3 (0.38) HTR1AHTR1DHTR1BNOS3NOS1
SCHEMBL7000439 0.68 SLC6A4 (0.42) HTR6HTR1AKDM4ELMNAPOLB
Oxalic Acid SCHEMBL7867378 0.67 SLC6A4 (0.52) HTR6SLC6A4
Bromide SCHEMBL7870832 0.65 SLC6A4 (0.57) HTR6HTR1AKDM4ELMNAPOLB
SCHEMBL6996625 0.64 SLC6A4 (0.62) HTR6HTR1AKDM4ELMNAPOLB
SCHEMBL8172220 0.62 QDPR (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003738-A1 BICYCLIC COMPOUNDS AS LIGANDS FOR 5-HT1 RECEPTORS SMITHKLINE BEECHAM PLC (GB) 2000-05-31 EP disclosed
WO-1999007700-A1 BICYCLIC COMPOUNDS AS LIGANDS FOR 5-HT1 RECEPTORS SMITHKLINE BEECHAM PLC (GB) 1999-02-18 WO disclosed