SCHEMBL8145398

SCHEMBL8145398

CC(C)(C)OC(=O)NCC[C@@]1(C(=O)OC(=O)OC(C)(C)C)CCCN1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GAA P10253 1/20 0.35
DRD2 P14416 5/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
CA12 O43570 4/20 0.32
CA1 P00915 4/20 0.32
CA2 P00918 4/20 0.32
CA9 Q16790 4/20 0.32
ALDH1A1 P00352 2/20 0.32
GFER P55789 1/20 0.32
TSHR P16473 1/20 0.31
ARG1 P05089 1/20 0.31
ARG2 P78540 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8149234 0.88 HCRTR2 (0.34) EPHX1TDP1MEN1KMT2AGAA
SCHEMBL7728931 0.88 HCRTR2 (0.34) EPHX1TDP1MEN1KMT2AGAA
SCHEMBL9637006 0.79 ARG1 (0.32) ARG1ARG2
SCHEMBL9730898 0.79 ARG1 (0.32) ARG1ARG2
SCHEMBL8135439 0.75 NPFFR1 (0.33) EPHX1TDP1MEN1KMT2AMAOA
SCHEMBL8150964 0.75 NPFFR1 (0.33) EPHX1TDP1MEN1KMT2AMAOA
SCHEMBL376992 0.73
SCHEMBL2497821 0.73
SCHEMBL8135118 0.73 P2RX7 (0.31) MEN1KMT2A
SCHEMBL7379886 0.72 HRH3 (0.46) CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed