SCHEMBL8146115

SCHEMBL8146115

CCc1cc(Nc2nc(N)c3ncn(CCO)c3n2)ccc1C

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.45
ADORA1 P30542 5/20 0.45
TMIGD3 P0DMS9 4/20 0.45
ADORA2B P29275 2/20 0.43
CDK1 P06493 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154514 0.79 ADORA2A (0.43) ADORA2AADORA1TMIGD3ADORA2BCDK1
SCHEMBL8153955 0.79 TK1 (0.58)
SCHEMBL5801330 0.73 HDAC3 (0.40)
SCHEMBL8158951 0.69 ADORA2A (0.40) ADORA2AADORA1TMIGD3ADORA2BCDK1
SCHEMBL19690966 0.68 CDK1 (0.45) CDK1
SCHEMBL12396113 0.68 TMIGD3 (0.41) ADORA2AADORA1TMIGD3ADORA2B
SCHEMBL8146043 0.67 CTSL (0.63) ADORA2AADORA1TMIGD3ADORA2BCDK1
SCHEMBL2160243 0.67 FGFR1 (0.47) ADORA2AADORA1TMIGD3ADORA2B
SCHEMBL8146595 0.67
SCHEMBL19691015 0.67 KCNN2 (0.51) CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772439-B1 Novel antibiotic compounds and antibiotic compositions comprising said compounds for inhibiting gram positive bacteria and mycoplasma cells. UNIV MASSACHUSETTS MEDICAL (US) 2000-10-04 EP claimed
EP-0772439-B1 Novel antibiotic compounds and antibiotic compositions comprising said compounds for inhibiting gram positive bacteria and mycoplasma cells. UNIV MASSACHUSETTS MEDICAL (US) 2000-10-04 EP disclosed
EP-0772439-A4 NOVEL ANTIBIOTIC COMPOUNDS AND METHODS TO TREAT GRAM-POSITIVE BACTERIAL AND MYCOPLASMAL INFECTIONS UNIV MASSACHUSETTS MEDICAL (US) 1998-01-07 EP disclosed
EP-0772439-A1 NOVEL ANTIBIOTIC COMPOUNDS AND METHODS TO TREAT GRAM-POSITIVE BACTERIAL AND MYCOPLASMAL INFECTIONS UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1997-05-14 EP disclosed
US-5516905-A ENZYME INHIBITORS OF DNA POLYMERASE FOR BACTERICIDES UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1996-05-14 US disclosed
WO-1996006614-A1 NOVEL ANTIBIOTIC COMPOUNDS AND METHODS TO TREAT GRAM-POSITIVE BACTERIAL AND MYCOPLASMAL INFECTIONS UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1996-03-07 WO disclosed