SCHEMBL8146809

SCHEMBL8146809

COC(=O)c1ccc(S(C)(=O)=O)c(-c2nnco2)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 1/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
KMT2A Q03164 3/20 0.35
HSD17B10 Q99714 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA12 O43570 1/20 0.34
TSHR P16473 1/20 0.33
VCAM1 P19320 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8132186 0.88 CA12 (0.36) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL8598024 0.81 CFTR (0.40) HSD17B10CA1CA2CA9VCAM1
SCHEMBL8164153 0.79 EDNRA (0.41) CYP3A4CYP2D6PSEN1PSEN2APH1B
SCHEMBL4273679 0.77 PSMB8 (0.38) HSD17B10ALDH1A1MAPTCA1CA2
SCHEMBL27561142 0.75 RAB9A (0.36) KMT2AHSD17B10ALDH1A1MAPTCA1
SCHEMBL4269505 0.75 SMN1; SMN2 (0.33) HSD17B10MAPTCA1CA2CA9
SCHEMBL8175098 0.75 GAA (0.42) KMT2AHSD17B10MAPTCA1CA2
SCHEMBL7946301 0.75 ACLY (0.44) KMT2AHSD17B10ALDH1A1MAPTCA1
SCHEMBL4274890 0.73 VCAM1 (0.33) CYP3A4CYP2D6KMT2AHSD17B10ALDH1A1
SCHEMBL8135182 0.73 MEN1 (0.41) KMT2AALDH1A1MAPTTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1104429-C 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides BASF AG (DE) 2003-04-02 CN disclosed
US-6165944-A 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides BASF AKTIENGESELLSCHAFT (DE) 2000-12-26 US disclosed
CN-1250447-A 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides BASF AG (DE) 2000-04-12 CN disclosed