SCHEMBL8148353

SCHEMBL8148353

CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)OCCCC(=O)OCI.CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)Oc1cccc(C(=O)O)c1CI

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
CTSL P07711 3/20 0.44
CTSS P25774 3/20 0.44
CTSB P07858 2/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 1/20 0.43
CTSK P43235 1/20 0.42
CASP3 P42574 2/20 0.39
CASP1 P29466 1/20 0.37
MME P08473 1/20 0.36
ECE1 P42892 1/20 0.36
KDM4E B2RXH2 1/20 0.36
RECQL P46063 1/20 0.36
REN P00797 1/20 0.35
ELANE P08246 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787420 0.91 CYP3A4 (0.38) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL3797250 0.90 CTSL (0.53) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL7676348 0.90 CTSL (0.53) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL7790304 0.87 CASP1 (0.36) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL3729686 0.86 CYP3A4 (0.58) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL3726928 0.82 CTSL (0.47) CTSLCTSSCTSBMEN1KMT2A
SCHEMBL3739436 0.81 CYP3A4 (0.62) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL3729516 0.79 CTSB (0.49) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL3740243 0.77 CYP3A4 (0.62) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A
SCHEMBL24131772 0.76 CTSB (0.48) CYP3A4CYP2D6CYP2C9CYP2C19RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054891-A1 PRODRUGS MEDIVIR AB (SE) 2000-11-29 EP disclosed
WO-1999041275-A1 PRODRUGS MEDIVIR AB (SE) 1999-08-19 WO disclosed