SCHEMBL8150757

SCHEMBL8150757

NC(=O)c1nc(Nc2ccc(Sc3ccccn3)c(Cl)c2)c2c[c]ncc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 2/20 0.38
ICAM1 P05362 1/20 0.36
SELE P16581 1/20 0.36
VCAM1 P19320 1/20 0.36
EGFR P00533 2/20 0.35
MAP2K1 Q02750 1/20 0.34
AURKA O14965 2/20 0.34
RPS6KB1 P23443 2/20 0.34
GRM4 Q14833 1/20 0.32
CSNK2A1 P68400 2/20 0.32
PIM1 P11309 1/20 0.32
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
KDR P35968 1/20 0.32
POLB P06746 1/20 0.32
ERBB2 P04626 2/20 0.32
ALDH1A1 P00352 1/20 0.32
PTPN11 Q06124 1/20 0.32
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487402 0.79 EGFR (0.30) EGFRCSNK2A1PIM1CSNK2A2CSNK2B
SCHEMBL2998232 0.79 EGFR (0.46) EGFRAURKARPS6KB1CSNK2A1CSNK2A2
SCHEMBL8490286 0.75 KMT2A (0.40) EGFRAURKARPS6KB1GRM4CSNK2A1
SCHEMBL2986229 0.73 AURKA (0.45) EGFRAURKARPS6KB1CSNK2A1KDR
SCHEMBL8082010 0.71 SYK (0.46) EGFRCSNK2A1KDRERBB2NPC1
SCHEMBL8096003 0.68 KDM4C (0.38) EGFRERBB2ALDH1A1
SCHEMBL8093494 0.68 XDH (0.33) KDRPOLBERBB2ALDH1A1NPC1
SCHEMBL8150759 0.68 GRM1 (0.61) EGFRERBB2
SCHEMBL4858939 0.67 AURKA (0.57) EGFRAURKARPS6KB1ERBB2
SCHEMBL4864883 0.67 AURKA (0.57) EGFRAURKARPS6KB1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127374-A AN ENZYME INHIBITOR FOR TREATING CANCER, RESTENOSIS, ATHEROSCLEROSIS, ENDOMETRIOSIS AND PSORIASIS WARNER-LAMBERT COMPANY (US) 2000-10-03 US disclosed