SCHEMBL8156987

SCHEMBL8156987

CCc1cccc(C=C(OCC(C)C)C(=O)c2cccc(OCC(C)C)c2OCC(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.39
ALDH1A1 P00352 2/20 0.39
AKR1C3 P42330 1/20 0.36
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
L3MBTL1 Q9Y468 4/20 0.33
MAPK1 P28482 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
HIF1A Q16665 1/20 0.33
MEN1 O00255 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
NPY1R P25929 1/20 0.32
NPY2R P49146 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MCL1 Q07820 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8159554 0.84 HTT (0.38) TSHRALDH1A1L3MBTL1MAPK1TDP1
SCHEMBL8158807 0.83 ALDH1A1 (0.38) TSHRALDH1A1AKR1C3L3MBTL1MAPK1
SCHEMBL8154299 0.82 ALOX5 (0.41) TSHRALDH1A1AKR1C3L3MBTL1MAPK1
SCHEMBL8145530 0.81 TSHR (0.42) TSHRALDH1A1L3MBTL1MAPK1TDP1
SCHEMBL8162733 0.81 ALDH1A1 (0.41) TSHRALDH1A1AKR1C3MEN1KMT2A
SCHEMBL8152762 0.80 TSHR (0.43) TSHRALDH1A1L3MBTL1MAPK1TDP1
SCHEMBL8153179 0.77 ABCB1 (0.42) TSHRL3MBTL1MEN1MAPTKMT2A
SCHEMBL8159015 0.77 KMT2A (0.39) TSHRALDH1A1AKR1C3L3MBTL1MAPK1
SCHEMBL8160025 0.76 AKR1C3 (0.37) TSHRALDH1A1AKR1C3L3MBTL1MAPK1
SCHEMBL8159064 0.75 PTGES (0.39) TSHRALDH1A1AKR1C3L3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996432-A2 BIOLOGICALLY ACTIVE 1,3-BIS-AROMATIC-PROP-2-EN-1-ONES, 1,3-BIS-AROMATIC-PROPAN-1-ONES, AND 1,3-BIS-AROMATIC-PROP-2-YN-1-ONES STATENS SERUMINSTITUT (DK) 2000-05-03 EP claimed
WO-1999000114-A2 BIOLOGICALLY ACTIVE 1,3-BIS-AROMATIC-PROP-2-EN-1-ONES, 1,3-BIS-AROMATIC-PROPAN-1-ONES, AND 1,3-BIS-AROMATIC-PROP-2-YN-1-ONES STATENS SERUM INSTITUT (DK) 1999-01-07 WO claimed