SCHEMBL8157747

SCHEMBL8157747

Cc1c(C)c(C)c2ccc[c]c2c1C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
HSP90AA1 P07900 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 2/20 0.31
CYP2A6 P11509 1/20 0.31
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28496768 0.86 CYP1A2 (0.33) NPC1HSP90AA1L3MBTL1CYP1A2CYP2A6
SCHEMBL15821385 0.73 MAOA (0.33) CYP1A2CYP2A6
SCHEMBL668081 0.71 CYP1A2 (0.48) L3MBTL1CYP1A2CYP2A6
SCHEMBL2409495 0.71 CYP2A6 (0.33) CYP1A2CYP2A6
SCHEMBL24104 0.69 HPRT1 (0.35) CYP1A2CYP2A6
SCHEMBL2407351 0.69 HPRT1 (0.35) CYP1A2CYP2A6
SCHEMBL4824194 0.69 HPRT1 (0.35) CYP1A2CYP2A6
SCHEMBL1556594 0.69 CYP1A2 (0.41) L3MBTL1CYP1A2CYP2A6AHR
SCHEMBL4584867 0.68 SMN1; SMN2 (0.36) NPC1L3MBTL1
SCHEMBL28986864 0.67 GPR3 (0.42) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0658585-B1 Aminophenylalanine derivatives, process for their production, their use and agents containing them as anti-coagulants STUEBER WERNER (DE) 2000-07-19 EP disclosed
CN-1039125-C Amidinophenylalanine derivatives and process for preparing same and use REHRINGWERKE AG (DE) 1998-07-15 CN disclosed
US-5571844-A Amidinophenylalanine derivatives, a process for their preparation, their use and compositions containing these as anticoagulants BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1996-11-05 US disclosed
EP-0513543-B1 Derivatives of amidinophenylalanine, procedure for their preparation, their utilisation and anticoagulant compositions comprising them. BEHRINGWERKE AG (DE) 1995-10-25 EP disclosed
EP-0658585-A2 Aminophenylalanine derivatives, process for their production, their use and agents containing them as anti-coagulants BEHRINGWERKE Aktiengesellschaft (DE) 1995-06-21 EP disclosed
CN-1067249-A Amidinophenylalaninederivatives derivatives and Preparation Method And The Use BEHRINGWERKE AG (DE) 1992-12-23 CN disclosed
EP-0513543-A1 Derivatives of amidinophenylalanine, procedure for their preparation, their utilisation and anticoagulant compositions comprising them. BEHRINGWERKE Aktiengesellschaft (DE) 1992-11-19 EP disclosed