SCHEMBL8158574

SCHEMBL8158574

COc1cccc(C=O)c1OCC(O)CN1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.61
DRD2 P14416 3/20 0.61
HTR1A P08908 2/20 0.61
ABCB11 O95342 1/20 0.52
CHRM2 P08172 1/20 0.52
ADRA2A P08913 1/20 0.52
CHRM1 P11229 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
DRD1 P21728 1/20 0.52
DRD4 P21917 1/20 0.52
ACHE P22303 1/20 0.52
SLC6A2 P23975 1/20 0.52
HTR2C P28335 1/20 0.52
SLC6A4 P31645 1/20 0.52
CCKBR P32239 1/20 0.52
ADRA1A P35348 1/20 0.52
HRH1 P35367 1/20 0.52
OPRM1 P35372 1/20 0.52
DRD3 P35462 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545277 0.85 HTR2A (0.61) HTR2ADRD2HTR1AABCB11CHRM2
SCHEMBL1545448 0.82 HTR2A (0.77) HTR2ADRD2HTR1AADRA2AACHE
SCHEMBL7977213 0.81 HTR2A (0.60) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL8888386 0.80 DRD2 (0.61) HTR2ADRD2HTR1AABCB11CHRM2
SCHEMBL7975053 0.80 HTR2A (0.64) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL1545018 0.78 DRD2 (0.72) HTR2ADRD2HTR1AACHESLC6A4
Hydrochloric Acid SCHEMBL1545656 0.78 ACHE (0.69) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL15703012 0.76 KCNH2 (0.74) HTR2ADRD2HTR1AKCNH2
SCHEMBL7974099 0.76 HTR2A (0.68) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL7974089 0.76 HTR2A (0.68) HTR2ADRD2HTR1AACHESLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6140345-A FOR TREATING PSYCHOSES AND PAIN AVENTIS PHARMACEUTICALS INC. 2000-10-31 US claimed