SCHEMBL8168501

SCHEMBL8168501

O=C(Cc1nnc(CCCNC2N=CCN2)s1)NC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.42
ITGAV P06756 6/20 0.42
ITGA2B P08514 17/20 0.41
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP12 P39900 1/20 0.36
MMP14 P50281 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8177319 0.92 ITGB3 (0.36) ITGB3ITGAVITGA2B
Hydrochloric Acid SCHEMBL8222330 0.91 ITGB3 (0.36) ITGB3ITGAVITGA2B
SCHEMBL8216110 0.85 F2 (0.33) ITGB3ITGA2B
SCHEMBL7366550 0.82 SLC1A2 (0.41)
SCHEMBL8168513 0.79 ITGB3 (0.53) ITGB3ITGAVITGA2B
SCHEMBL8168330 0.76 ITGAV (0.44) ITGB3ITGAVITGA2B
SCHEMBL7367606 0.75 SLC1A3 (0.36)
Hydrochloric Acid SCHEMBL8215964 0.75 GLS (0.33)
SCHEMBL8176077 0.73 ITGAV (0.46) ITGB3ITGAVITGA2B
SCHEMBL8218077 0.73 GLS (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153628-A 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists DUPONT PHARMACEUTICALS COMPANY (US) 2000-11-28 US disclosed