SCHEMBL7367606

SCHEMBL7367606

Cc1cccc(S(=O)(=O)NC(C(=O)O)C(N)C(=O)Cc2nnc(CCCN[C@@H]3N=CCN3)s2)c1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 9/20 0.36
SLC1A2 P43004 9/20 0.36
SLC1A1 P43005 8/20 0.36
GLS O94925 2/20 0.34
F2 P00734 2/20 0.32
ALDH1A1 P00352 1/20 0.32
FBP1 P09467 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366550 0.92 SLC1A2 (0.41) SLC1A3SLC1A2SLC1A1GLS
SCHEMBL8177319 0.84 ITGB3 (0.36) GLSF2FBP1
Hydrochloric Acid SCHEMBL8222330 0.84 ITGB3 (0.36) GLSF2FBP1
SCHEMBL8216110 0.80 F2 (0.33) GLSF2FBP1
SCHEMBL7366853 0.76 SLC1A3 (0.34) SLC1A3SLC1A2SLC1A1
SCHEMBL8168501 0.75 ITGB3 (0.42)
Hydrochloric Acid SCHEMBL8215964 0.75 GLS (0.33) GLS
SCHEMBL8218077 0.75 GLS (0.33) GLS
SCHEMBL7367243 0.73 SLC1A3 (0.47) SLC1A3SLC1A2SLC1A1F2ALDH1A1
SCHEMBL8176077 0.65 ITGAV (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1049693-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS $g(a) v?$g(b) 3? ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-08 EP claimed
WO-1999026945-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS αvβ3 ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-06-03 WO claimed
EP-1049693-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS $g(a) v?$g(b) 3? ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-08 EP disclosed
WO-1999026945-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS αvβ3 ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-06-03 WO disclosed