SCHEMBL8170649

SCHEMBL8170649

CC(=O)N1CCCC(n2c(C3=CCCC=C3)c(C(=O)N3CCNCC3)n(CCCNS(=O)(=O)c3ccccc3)c2=O)C1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
HTR7 P34969 1/20 0.31
CNR2 P34972 1/20 0.30
HTR2A P28223 1/20 0.30
TMEM97 Q5BJF2 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL884696 0.90 POLB (0.34) ALDH1A1POLBPKMHTR7CNR2
SCHEMBL885714 0.85 POLB (0.35) ALDH1A1POLBPKMHTR2ATMEM97
SCHEMBL884541 0.80 CYP2C19 (0.36) ALDH1A1PKM
SCHEMBL886810 0.80 CTSK (0.33) CNR2
SCHEMBL8174751 0.78 ACP1 (0.37) ALDH1A1PKMHTR7
SCHEMBL884768 0.77 SLC6A2 (0.38) ALDH1A1SIGMAR1
SCHEMBL885599 0.76 HDAC1 (0.33) ALDH1A1
SCHEMBL8169739 0.76 SIGMAR1 (0.36) CNR2HTR2ATMEM97SIGMAR1
SCHEMBL884320 0.75 LMNA (0.39) ALDH1A1PKM
SCHEMBL885631 0.75 CTSK (0.33) HTR7HTR2ATMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089005-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-07-24 WO disclosed