SCHEMBL8172016

SCHEMBL8172016

c1ccc(N2CCN(Cc3nsc(N4CCN(c5ccccn5)CC4)n3)CC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
KDM4E B2RXH2 5/20 0.53
TDP1 Q9NUW8 1/20 0.53
DRD4 P21917 4/20 0.51
DRD2 P14416 2/20 0.51
CYP3A4 P08684 1/20 0.50
ALOX15 P16050 1/20 0.50
OPRK1 P41145 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
GRM2 Q14416 1/20 0.50
MAPK1 P28482 4/20 0.48
TSHR P16473 1/20 0.48
USP2 O75604 1/20 0.48
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.48
HTT P42858 2/20 0.48
RAB9A P51151 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
SORD Q00796 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8163279 0.84 MAPT (0.48) ALDH1A1KDM4ETDP1MAPK1NPC1
SCHEMBL8558421 0.78 ALDH1A1 (0.55) ALDH1A1KDM4ETDP1DRD4DRD2
SCHEMBL8170319 0.78 MAPT (0.52) ALDH1A1KDM4EMAPK1TSHRNPC1
SCHEMBL8170423 0.76 FAAH (0.61) ALDH1A1MAPK1NPC1MAPTHTT
SCHEMBL8169372 0.75 HTT (0.49) ALDH1A1KDM4ECYP3A4MAPK1TSHR
SCHEMBL12858870 0.74 ALDH1A1 (0.62) ALDH1A1KDM4ETDP1DRD4DRD2
SCHEMBL30936089 0.74 ALDH1A1 (0.62) ALDH1A1KDM4ETDP1DRD4DRD2
SCHEMBL8111511 0.74 HTT (0.77) ALDH1A1KDM4ETDP1DRD4DRD2
SCHEMBL15190465 0.73 MEN1 (0.41) ALDH1A1KDM4EMAPK1NPC1MAPT
SCHEMBL13711971 0.73 KCNH2 (0.71) ALDH1A1DRD4DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6060472-A Thiadiazole compounds useful as inhibitors of H+ /K+ atpase APOTEX INC. (CA) 2000-05-09 US claimed
WO-1999051584-A1 THIADIAZOLE COMPOUNDS USEFUL AS INHIBITORS OF H+/K+ ATPASE APOTEX INC. (CA) 1999-10-14 WO claimed