SCHEMBL8558421

SCHEMBL8558421

c1ccc(N2CCN(Cc3ncsn3)CC2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
KDM4E B2RXH2 5/20 0.55
TDP1 Q9NUW8 1/20 0.55
DRD4 P21917 4/20 0.50
MAPT P10636 3/20 0.50
DRD2 P14416 2/20 0.50
HTT P42858 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 2/20 0.49
DRD3 P35462 1/20 0.49
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
OPRK1 P41145 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
GRM2 Q14416 1/20 0.49
POLB P06746 1/20 0.49
KCNH2 Q12809 1/20 0.49
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556657 0.82 MEN1 (0.51) ALDH1A1KDM4EDRD4DRD2KMT2A
SCHEMBL8555562 0.81 DRD4 (0.54) ALDH1A1KDM4EDRD4MAPTDRD2
SCHEMBL8489945 0.79 PLD1 (0.53) ALDH1A1KDM4EMAPTHTTNPC1
SCHEMBL8172016 0.78 ALDH1A1 (0.53) ALDH1A1KDM4ETDP1DRD4MAPT
SCHEMBL8556503 0.78 SIGMAR1 (0.58) ALDH1A1DRD4DRD2KMT2ADRD3
SCHEMBL8111511 0.76 HTT (0.77) ALDH1A1KDM4ETDP1DRD4MAPT
SCHEMBL30936089 0.76 ALDH1A1 (0.62) ALDH1A1KDM4ETDP1DRD4MAPT
SCHEMBL12858870 0.76 ALDH1A1 (0.62) ALDH1A1KDM4ETDP1DRD4MAPT
SCHEMBL13711971 0.75 KCNH2 (0.71) ALDH1A1DRD4DRD2DRD3POLB
SCHEMBL15800694 0.74 PLD1 (0.73) ALDH1A1KDM4EMAPTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP claimed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO claimed
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP disclosed
EP-0883606-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1998-12-16 EP disclosed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO disclosed
WO-1997031893-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1997-09-04 WO disclosed