SCHEMBL9511093

SCHEMBL9511093

CC(C)(C)N(NC(=O)c1ccc(F)cc1)C(=O)c1ccccn1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
POLB P06746 1/20 0.55
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
RECQL P46063 1/20 0.48
CES1 P23141 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8173935 0.90 POLB (0.55) AGTR1NPC1RAB9APOLBMEN1
SCHEMBL8173237 0.90 POLB (0.68) POLBKMT2ACYP3A4CYP2C9
SCHEMBL9815800 0.89 POLB (0.56) POLBMEN1KMT2ACYP3A4CYP2C9
SCHEMBL9425189 0.85 HPGD (0.68) POLBCYP3A4CYP2C9
SCHEMBL9425890 0.85 TLR7 (0.64) NPC1RAB9APOLBMEN1KMT2A
SCHEMBL9815864 0.82 ABCB1 (0.60) POLBCYP3A4CYP2C9
SCHEMBL9509589 0.82 MEN1 (0.57) NPC1RAB9APOLBMEN1KMT2A
SCHEMBL9815896 0.82 GRM4 (0.55)
SCHEMBL8773661 0.81 POLB (0.82) POLBCYP3A4CYP2C9RECQL
SCHEMBL8773658 0.81 POLB (0.82) POLBCYP3A4CYP2C9RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed