SCHEMBL9815864

SCHEMBL9815864

Cc1cc(C)cc(C(=O)NN(C(=O)c2ccccn2)C(C)(C)C)c1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 7/20 0.60
CYP3A4 P08684 2/20 0.53
POLB P06746 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9425270 0.90 ABCB1 (0.64) ABCB1CYP3A4POLBCYP2C9
SCHEMBL9815800 0.89 POLB (0.56) ABCB1CYP3A4POLBCYP2C9
SCHEMBL8173237 0.87 POLB (0.68) CYP3A4POLBCYP2C9
SCHEMBL9425963 0.83 ABCB1 (0.64) ABCB1CYP3A4POLBCYP2C9
SCHEMBL9511093 0.82 AGTR1 (0.55) CYP3A4POLBCYP2C9
SCHEMBL9509589 0.82 MEN1 (0.57) ABCB1CYP3A4POLBCYP2C9
SCHEMBL9511092 0.81 POLB (0.77) ABCB1CYP3A4POLBCYP2C9
SCHEMBL9426147 0.81 POLB (0.56) ABCB1CYP3A4POLBCYP2C9
SCHEMBL9425189 0.81 HPGD (0.68) ABCB1CYP3A4POLBCYP2C9
SCHEMBL9815793 0.80 ABCB1 (0.62) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed