SCHEMBL8174331

SCHEMBL8174331

NC(=O)c1cnccc1-n1cccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT3 Q9NTG7 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
CYP46A1 Q9Y6A2 1/20 0.46
IRAK4 Q9NWZ3 2/20 0.44
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
G6PD P11413 1/20 0.42
KMT2A Q03164 1/20 0.42
ATR Q13535 1/20 0.41
SYK P43405 1/20 0.41
TDO2 P48775 1/20 0.41
HTT P42858 1/20 0.40
F7 P08709 1/20 0.39
F3 P13726 1/20 0.39
SARM1 Q6SZW1 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30298688 0.88 CYP46A1 (0.46) SIRT3TDP1CYP46A1IRAK4KDM4E
SCHEMBL7090853 0.86 LMNA (0.48) TDP1CYP46A1KDM4ELMNAALDH1A1
SCHEMBL3544059 0.82 NPC1 (0.49) IRAK4KDM4ELMNAALDH1A1MEN1
SCHEMBL21816147 0.81 ALDH1A1 (0.48) CYP46A1KDM4ELMNAALDH1A1MEN1
SCHEMBL885410 0.79 SIRT3 (0.49) SIRT3TDP1IRAK4KDM4ELMNA
SCHEMBL7848026 0.78 HCRTR1 (0.48) SIRT3TDP1IRAK4KDM4ESYK
SCHEMBL16666154 0.76 NOTUM (0.46) KDM4ELMNAALDH1A1MEN1GAA
SCHEMBL15771021 0.75 TDO2 (0.50) TDP1CYP46A1KDM4ELMNAALDH1A1
SCHEMBL2732235 0.74 CSF1R (0.44) SIRT3IRAK4SYKSIRT2SIRT1
SCHEMBL8174469 0.74 CTNNB1 (0.40) SIRT3CYP46A1KDM4ELMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925322-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2015-10-07 EP claimed
CN-102933548-B Carboxamide compounds and their use as calpain inhibitors ABBOTT LAB 2015-03-11 CN claimed
WO-2014085210-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2014-06-05 WO claimed
WO-2000031066-A1 SUBSTITUTED N-PYRAZOLYL-PHENOXYNICOTINIC ACID-(THIO)AMIDES THAT CAN BE USED AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2000-06-02 WO claimed
CN-102933548-B Carboxamide compounds and their use as calpain inhibitors ABBOTT LAB 2015-03-11 CN disclosed
WO-2000031066-A1 SUBSTITUTED N-PYRAZOLYL-PHENOXYNICOTINIC ACID-(THIO)AMIDES THAT CAN BE USED AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2000-06-02 WO disclosed