SCHEMBL8174337

SCHEMBL8174337

COC(=O)c1coc(CC(NC(=O)OC(C)(C)C)c2ccc(F)cc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 5/20 0.46
KCNH2 Q12809 2/20 0.46
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
TSHR P16473 3/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ALDH1A1 P00352 4/20 0.36
NPSR1 Q6W5P4 3/20 0.36
TP53 P04637 2/20 0.36
HPGD P15428 2/20 0.36
HTT P42858 2/20 0.36
HSD17B10 Q99714 2/20 0.36
JAK2 O60674 1/20 0.36
MAPK1 P28482 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5014183 0.90 SLC6A2 (0.46) CACNA1GCTSSCTSKTSHRLMNA
SCHEMBL8174332 0.82 ALDH1A1 (0.46) CTSSCTSKTSHRLMNAMEN1
SCHEMBL8174330 0.82 ALDH1A1 (0.46) CTSSCTSKTSHRLMNAMEN1
SCHEMBL5014055 0.81 CTSK (0.43) CTSSCTSKTSHRLMNAMEN1
SCHEMBL8184215 0.81 TSHR (0.41) CTSSCTSKTSHRLMNAMEN1
SCHEMBL1196722 0.79 ACE (0.45) CTSSCTSKSLC6A2SLC6A4SLC6A3
SCHEMBL7615051 0.76 TSHR (0.43) CTSSCTSKTSHRLMNAMEN1
SCHEMBL5013656 0.74 PCSK9 (0.46) CACNA1GKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL12980639 0.74 C3AR1 (0.46) CTSKTSHRLMNAMEN1KMT2A
SCHEMBL10045822 0.74 C3AR1 (0.46) CTSKTSHRLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156732-A Azole peptidomimetics as thrombin receptor antagonists ORTHO-MCNEIL PHARMACEUTICALS, INC. (US) 2000-12-05 US disclosed
US-6017890-A Azole peptidomimetics as thrombin receptor antagonists ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-01-25 US disclosed