SCHEMBL5014183

SCHEMBL5014183

COC(=O)c1coc(CC(NC(=O)OC(C)(C)C)c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
CACNA1G O43497 2/20 0.44
ALDH1A1 P00352 3/20 0.42
CTSS P25774 3/20 0.42
CTSK P43235 2/20 0.42
NPSR1 Q6W5P4 3/20 0.41
TSHR P16473 3/20 0.41
LMNA P02545 2/20 0.41
PKM P14618 2/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 2/20 0.41
HSD17B10 Q99714 2/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
AGTR1 P30556 1/20 0.41
RAB9A P51151 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5014055 0.91 CTSK (0.43) ALDH1A1CTSSCTSKNPSR1TSHR
SCHEMBL8174337 0.90 CACNA1G (0.46) SLC6A2SLC6A4SLC6A3CACNA1GALDH1A1
SCHEMBL1196722 0.83 ACE (0.45) SLC6A2SLC6A4SLC6A3CTSSCTSK
SCHEMBL5014182 0.81 ALDH1A1 (0.56) ALDH1A1CTSSCTSKNPSR1TSHR
SCHEMBL16763402 0.78 CHRM3 (0.56) SLC6A2SLC6A4SLC6A3CACNA1G
SCHEMBL16763400 0.78 CHRM3 (0.56) SLC6A2SLC6A4SLC6A3CACNA1G
SCHEMBL7735821 0.77 MAPT (0.47) ALDH1A1CTSSCTSKNPSR1TSHR
SCHEMBL5013656 0.76 PCSK9 (0.46) SLC6A2SLC6A4SLC6A3CACNA1GNPSR1
SCHEMBL801072 0.76 PPARA (0.51) ALDH1A1CTSSNPSR1TSHRLMNA
SCHEMBL12980639 0.75 C3AR1 (0.46) ALDH1A1CTSKNPSR1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009942-A1 HETEROAROMATIC-BASED PEPTIDE MACROCYCLES AS G-QUADRUPLEX LIGANDS CAMBRIDGE ENTERPRISE LTD. (GB) 2008-01-24 WO disclosed