SCHEMBL8174459

SCHEMBL8174459

NC(=O)c1c(O)cccc1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.54
CES1 P23141 2/20 0.54
CA12 O43570 4/20 0.48
CA1 P00915 4/20 0.48
CA2 P00918 4/20 0.48
CA7 P43166 4/20 0.48
CA9 Q16790 4/20 0.48
CA14 Q9ULX7 4/20 0.48
THRB P10828 1/20 0.46
PARP1 P09874 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
SPR P35270 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL203321 0.86 CES2 (0.64) CES2CES1PARP1MEN1KMT2A
Hydrochloric Acid SCHEMBL5053757 0.84 CES2 (0.61) CES2CES1PARP1MEN1KMT2A
SCHEMBL28267101 0.84 CES2 (0.61) CES2CES1PARP1MEN1KMT2A
SCHEMBL1668962 0.84 CA2 (0.59) CA12CA1CA2CA7CA9
SCHEMBL23463704 0.83 PARP1 (0.47) CES2CES1CA12CA1CA2
SCHEMBL617480 0.80 CA12 (0.70) CES2CES1CA12CA1CA2
SCHEMBL29349853 0.78 CES2 (0.54) CES2CES1PARP1KDM4EALDH1A1
SCHEMBL164708 0.78 CES2 (0.54) CES2CES1PARP1MEN1KMT2A
SCHEMBL28871108 0.78 CA12 (0.67) CES2CES1CA12CA1CA2
SCHEMBL11266406 0.78 CES2 (0.54) CES2CES1PARP1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624567-A2 Derivatives of 3-fluorophenol, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-17 EP claimed
CN-105263901-A [alpha]-substituted glycineamide derivative KISSEI PHARMACEUTICAL 2016-01-20 CN disclosed
US-6100246-A Spiro-piperidine derivatives as inhibitors of nitric oxide synthase ASTRA PHARMACEUTICALS LIMITED (GB) 2000-08-08 US disclosed
CN-1259132-A Compounds ASTRA PHARMA PROD (GB) 2000-07-05 CN disclosed
EP-0975639-A1 COMPOUNDS Astra Pharmaceuticals Limited (GB) 2000-02-02 EP disclosed
WO-1998046611-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-10-22 WO disclosed
EP-0624567-A2 Derivatives of 3-fluorophenol, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-17 EP disclosed