SCHEMBL8176181

SCHEMBL8176181

COC(=O)C(CNC(=O)Cc1nnc(CCC[N+](=O)[O-])s1)NS(=O)(=O)c1cccc(C)c1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.37
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
KMT2A Q03164 1/20 0.36
F2 P00734 4/20 0.35
FBP1 P09467 10/20 0.35
ITGAV P06756 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8176184 1.00 GLS (0.37) GLSMEN1CYP3A4MAPTCYP2C9
SCHEMBL8210927 0.89 F2 (0.40) GLSMEN1CYP3A4MAPTCYP2C9
SCHEMBL8210925 0.89 F2 (0.40) GLSMEN1CYP3A4MAPTCYP2C9
SCHEMBL8216119 0.81 ITGB3 (0.39) GLSF2ITGAV
SCHEMBL8216110 0.80 F2 (0.33) GLSMEN1CYP3A4MAPTCYP2C9
SCHEMBL8177325 0.73 ITGB3 (0.46) F2ITGAV
SCHEMBL8177319 0.72 ITGB3 (0.36) GLSF2FBP1ITGAV
Hydrochloric Acid SCHEMBL8222330 0.72 ITGB3 (0.36) GLSF2FBP1ITGAV
SCHEMBL8167396 0.69 GLS (0.38) GLS
SCHEMBL7379009 0.67 KMT2A (0.49) KMT2AF2FBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153628-A 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists DUPONT PHARMACEUTICALS COMPANY (US) 2000-11-28 US disclosed