SCHEMBL8177205

SCHEMBL8177205

CC(C)c1cc(C#N)cc(C(C)C)c1OS(N)(=O)=O

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.46
CA2 P00918 7/20 0.46
CA9 Q16790 7/20 0.46
STS P08842 2/20 0.38
CA12 O43570 2/20 0.36
CYP19A1 P11511 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27561893 0.81 GABRA1 (0.44) CA1CA2CA9CA12
SCHEMBL8898620 0.80 CA1 (0.50) CA1CA2CA9STSCA12
SCHEMBL8175444 0.80 CA2 (0.39) CA1CA2CA9STSCA12
SCHEMBL27564440 0.79 CA2 (0.41) CA1CA2CA9CA12
SCHEMBL8495954 0.79 FABP4 (0.48) CA1CA2CA9CA12
SCHEMBL27561891 0.77 CA2 (0.45) CA1CA2CA9
SCHEMBL27582518 0.77 CA2 (0.58) CA1CA2CA9CA12
SCHEMBL27561967 0.77 CA1 (0.40) CA1CA2CA9CA12
SCHEMBL11791229 0.77 FABP4 (0.39) CA1CA2CA9CA12
SCHEMBL27561904 0.76 CA2 (0.48) CA1CA2CA9STSCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6093744-A USE AS CEREBROVASCULAR AGENTS IN DISEASES SUCH AS STROKE, PERIPHERAL VASCULAR DISEASE, RESTENOSIS, AND AS AGENTS FOR REGULATING PLASMA CHOLESTEROL CONCENTRATIONS, FOR TREATING HYPERCHOLESTEROLEMIA AND ATHEROSCLEROSIS WARNER-LAMBERT COMPANY (US) 2000-07-25 US disclosed