SCHEMBL8180809

SCHEMBL8180809

CC(C)=CCN(C(=O)OC(C)(C)C)c1cc(OCc2ccccc2)c2ccc(C#N)cc2c1Br

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.36
CYP19A1 P11511 1/20 0.36
CACNA1B Q00975 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
ABCB1 P08183 1/20 0.34
PDCD1 Q15116 6/20 0.34
CD274 Q9NZQ7 6/20 0.34
NCEH1 Q6PIU2 1/20 0.34
PTGER1 P34995 1/20 0.34
PPIA P62937 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
SLC6A9 P48067 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8197532 0.92 MRGPRX4 (0.38) MRGPRX4CYP19A1CYP11B1CYP11B2ABCB1
SCHEMBL8321897 0.86 MTNR1A (0.40) CACNA1B
SCHEMBL8132245 0.82 MRGPRX4 (0.36) MRGPRX4CYP19A1CYP11B1CYP11B2ABCB1
SCHEMBL8191113 0.81 PTGER1 (0.33) MRGPRX4CYP19A1CYP11B1CYP11B2ABCB1
SCHEMBL8317086 0.78 HDAC8 (0.40)
SCHEMBL8190897 0.76 MRGPRX4 (0.40) MRGPRX4CYP19A1PTGER1PPIAMAOB
SCHEMBL14502597 0.74 GLRA1 (0.35) MRGPRX4CYP19A1PTGER1MAOB
SCHEMBL8131442 0.74 MRGPRX4 (0.39) MRGPRX4CACNA1B
SCHEMBL7953762 0.73 L3MBTL1 (0.38) MRGPRX4PTGER1
SCHEMBL8127756 0.73 MRGPRX4 (0.40) MRGPRX4CYP19A1CYP11B1CYP11B2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6060608-A ANTITUMOR AGENTS THE SCRIPPS RESEARCH INSTITUTE (US) 2000-05-09 US disclosed