SCHEMBL8317086

SCHEMBL8317086

COc1ccc2c(OCc3ccccc3)cc(N(CC=O)C(=O)OC(C)(C)C)c(Br)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.40
MTNR1A P48039 3/20 0.39
MTNR1B P49286 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
APP P05067 2/20 0.39
SLC2A1 P11166 1/20 0.38
LRRK2 Q5S007 1/20 0.37
KDM4E B2RXH2 2/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
TLR9 Q9NR96 2/20 0.37
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
RECQL P46063 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8321897 0.91 MTNR1A (0.40) HDAC8MTNR1AMTNR1BL3MBTL1APP
SCHEMBL8197532 0.86 MRGPRX4 (0.38)
SCHEMBL7953762 0.79 L3MBTL1 (0.38) L3MBTL1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL8180809 0.78 MRGPRX4 (0.36)
SCHEMBL6205852 0.77 CYP2C9 (0.46) HDAC8MTNR1AMTNR1BLRRK2KDM4E
SCHEMBL8132061 0.76 MRGPRX4 (0.40) L3MBTL1NPC1GAARAB9ASMN1; SMN2
SCHEMBL7952320 0.75 L3MBTL1 (0.42) L3MBTL1APPKDM4EPOLBNPSR1
SCHEMBL7959955 0.73 L3MBTL1 (0.35) HDAC8MTNR1AMTNR1BL3MBTL1APP
SCHEMBL6324123 0.73 L3MBTL1 (0.40) L3MBTL1APPKDM4ETLR9NPSR1
SCHEMBL13311249 0.72 L3MBTL1 (0.37) L3MBTL1SMN1; SMN2KEAP1NFE2L2TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985908-A MCBI (7-METHOXY-1,2,9A-TETRA-HYDROCYCLOPROPA(C)BENZ(E)INDOL-4-ONE) IS EMPLOYABLE AS A DNA ALKYLATING AGENT AND CAN BE INCORPORATED INTO ANALOGS OF CC-1065 AND THE DUOCARMYCINS FOR THE SCRIPPS RESEARCH INSTITUTE (US) 1999-11-16 US disclosed