SCHEMBL8181122

SCHEMBL8181122

O=C(O)Cc1ccc2occcc1-2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.41
PTPN1 P18031 4/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
KEAP1 Q14145 1/20 0.37
SRC P12931 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
PTPN2 P17706 1/20 0.36
PTPN6 P29350 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5665316 0.91 AKR1B1 (0.48) AKR1B1PTPN1PTGDR2SMN1; SMN2TDP1
SCHEMBL1282584 0.84 CYP2C19 (0.38) PTPN1ALOX15TDP1CYP2C19ALDH1A1
SCHEMBL9550467 0.84 PTPN1 (0.37) PTPN1ALOX15TDP1KEAP1TSHR
SCHEMBL8382068 0.81 KEAP1 (0.51) PTPN1MAPTSMN1; SMN2TDP1KEAP1
SCHEMBL5546711 0.77 SLC9A1 (0.40) PTPN1MAPTALOX15TDP1L3MBTL1
SCHEMBL2095737 0.75 KDM4E (0.37) PTPN1MAPTALOX15TDP1TSHR
SCHEMBL21767386 0.72 OPRM1 (0.43) MAPTALOX15SMN1; SMN2TDP1TSHR
SCHEMBL7827157 0.72 AKR1B1 (0.67) AKR1B1MAPTTDP1TSHR
SCHEMBL4141035 0.72 PTPN1 (0.51) PTPN1MAPTALOX15TDP1KEAP1
SCHEMBL4649113 0.72 AKR1B1 (0.50) AKR1B1PTPN1MAPTTDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057357-A USEFUL IN TREATING PAIN, INFLAMMATION, PSORIASIS AND IRRITABLE BOWEL SYNDROME WARNER-LAMBERT COMPANY (US) 2000-05-02 US disclosed
WO-1998049158-A1 PERIPHERALLY SELECTIVE KAPPA OPIOID AGONISTS WARNER-LAMBERT COMPANY (US) 1998-11-05 WO disclosed
EP-0552386-A1 2-Amino-3 or 6-methoxycyclohexyl amide derivatives WARNER-LAMBERT COMPANY (US) 1993-07-28 EP disclosed
US-5051428-A 2-amino-4 or 5-methoxycyclohexyl amides useful as analgesics WARNER-LAMBERT COMPANY (US) 1991-09-24 US disclosed
EP-0372466-A2 2-Amino-4 or 5-methoxycyclohexyl amides useful as analgesics WARNER-LAMBERT COMPANY (US) 1990-06-13 EP disclosed