SCHEMBL8181685

SCHEMBL8181685

NC1CCC(n2c(=O)c3cc(F)cnc3n(-c3cccc(-c4ccc(CN5CCN(C6CCCC6)CC5)cc4)c3)c2=O)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.37
TSHR P16473 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
DRD3 P35462 2/20 0.35
PDE4B Q07343 1/20 0.34
CDK1 P06493 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
TNF P01375 1/20 0.34
LITAF Q99732 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL870966 1.00 METAP2 (0.37) METAP2TSHRNPSR1CRHBPCRHR2
SCHEMBL870965 1.00 METAP2 (0.37) METAP2TSHRNPSR1CRHBPCRHR2
SCHEMBL871727 0.94 PDE4B (0.39) METAP2TSHRNPSR1CRHBPCRHR2
SCHEMBL872430 0.90 CHKA (0.41)
SCHEMBL871025 0.90 CHKA (0.41)
SCHEMBL870887 0.90 VCP (0.37) TSHRNPSR1CRHBPCRHR2SMN1; SMN2
SCHEMBL870886 0.90 VCP (0.37) TSHRNPSR1CRHBPCRHR2SMN1; SMN2
SCHEMBL870187 0.89 PDE4B (0.41) TSHRNPSR1CRHBPCRHR2SMN1; SMN2
SCHEMBL870188 0.89 PDE4B (0.41) TSHRNPSR1CRHBPCRHR2SMN1; SMN2
SCHEMBL3029957 0.89 PDE4B (0.43) ALDH1A1MEN1KMT2ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008084223-A2 CHEMICAL COMPOUNDS 637: PYRIDOPYRIMIDINEDIONES AS PDE4 INHIBITORS ASTRAZENECA AB (SE) 2008-07-17 WO disclosed