SCHEMBL8184169

SCHEMBL8184169

COc1ccc2c(O)cc(=O)n(C)c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
MAPT P10636 4/20 0.59
KDM4E B2RXH2 3/20 0.59
HPGD P15428 3/20 0.59
HSD17B10 Q99714 3/20 0.59
THRB P10828 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
EGFR P00533 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAOA P21397 3/20 0.44
DYRK1A Q13627 1/20 0.44
CA2 P00918 1/20 0.43
SRC P12931 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30507409 1.00 ALDH1A1 (0.59) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL6208739 0.87 MAPT (0.56) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL392780 0.82 NQO2 (0.57) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL29857369 0.82 KDM4E (0.54) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL29889991 0.81 KDM4E (0.52) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL30507425 0.81 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL28513249 0.81 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL6608635 0.78 AR (0.47) ALDH1A1KDM4EHPGDHSD17B10EGFR
SCHEMBL18288081 0.78 L3MBTL1 (0.60) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL11825468 0.77 ALDH1A1 (0.62) ALDH1A1MAPTKDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-B Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2023-07-25 CN disclosed
CN-112010844-A Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2020-12-01 CN disclosed
US-6143766-A ENZYME INHIBITORS WITH IMIDAZOLE GROUPS WARNER-LAMBERT COMPANY (US) 2000-11-07 US disclosed