SCHEMBL28513249

SCHEMBL28513249

COc1ccc2c(Cl)cc(=O)n(C)c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 5/20 0.46
HPGD P15428 4/20 0.46
HSD17B10 Q99714 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 2/20 0.46
GLA P06280 1/20 0.46
EGFR P00533 1/20 0.45
MAOA P21397 3/20 0.44
DYRK1A Q13627 1/20 0.44
MAPT P10636 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
GRM2 Q14416 1/20 0.41
MAPK14 Q16539 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
APAF1 O14727 1/20 0.41
PABPC1 P11940 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30507425 1.00 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL829534 0.87 MAPT (0.53) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL392780 0.82 NQO2 (0.57) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL8184169 0.81 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL30507409 0.81 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL30727441 0.80 MAT2A (0.50) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL6608635 0.78 AR (0.47) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL18288081 0.78 L3MBTL1 (0.60) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL30507475 0.77 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL28497698 0.77 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-B Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2023-07-25 CN disclosed
CN-112010844-A Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2020-12-01 CN disclosed