SCHEMBL8190644

SCHEMBL8190644

COc1cccc(/C=C/C2=NN=C(C)Cc3cc4c(cc32)OCO4)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.44
CYP1A1 P04798 3/20 0.44
CYP1B1 Q16678 3/20 0.44
MAPT P10636 4/20 0.43
KMT2A Q03164 3/20 0.43
CYP2D6 P10635 2/20 0.43
MEN1 O00255 2/20 0.43
NFKB1 P19838 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
GRIA2 P42262 1/20 0.43
HIF1A Q16665 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.43
NFE2L2 Q16236 5/20 0.42
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 1/20 0.40
NPC1 O15118 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8190647 1.00 CYP1A2 (0.44) CYP1A2CYP1A1CYP1B1MAPTKMT2A
Hydrochloric Acid SCHEMBL9068728 0.99 LMNA (0.44) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL8184028 0.83 ALDH1A1 (0.47) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL8184031 0.83 ALDH1A1 (0.47) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL8191021 0.82 CYP1A2 (0.46) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL8191019 0.82 CYP1A2 (0.46) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL7993615 0.82 KDM4E (0.46) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL7993617 0.82 KDM4E (0.46) CYP1A2CYP1A1CYP1B1MAPTKMT2A
SCHEMBL8345585 0.79 MEN1 (0.47) CYP1A2MAPTKMT2ACYP2D6MEN1
SCHEMBL8345582 0.79 MEN1 (0.47) CYP1A2MAPTKMT2ACYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6075018-A TRANQUILIZERS EGIS GYOGYSZERGYAR RT. (HU) 2000-06-13 US disclosed