SCHEMBL8190802

SCHEMBL8190802

Cn1c(C(F)(F)F)cnc(-c2ccc(Cl)cc2Cl)c1=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.44
ALDH1A1 P00352 2/20 0.43
F2RL3 Q96RI0 1/20 0.40
TNKS O95271 1/20 0.39
CNR1 P21554 5/20 0.39
CNR2 P34972 4/20 0.39
DPP4 P27487 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
CRHR1 P34998 1/20 0.37
COMT P21964 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8179014 0.88 HSD11B1 (0.45) HSD11B1ALDH1A1TNKSCOMTHSD17B10
SCHEMBL8178803 0.81 COMT (0.34) ALDH1A1COMTKDM4E
SCHEMBL8187079 0.81 COMT (0.41) ALDH1A1L3MBTL1COMT
SCHEMBL8192289 0.79 HSP90AA1 (0.36) ALDH1A1COMTHSD17B10
SCHEMBL8177447 0.78 AKR1B1 (0.37) HSD11B1ALDH1A1KDM4EHPGD
SCHEMBL8188251 0.77 MAPK14 (0.43) ALDH1A1HSD17B10
SCHEMBL8177457 0.76 ALDH1A1 (0.33) HSD11B1ALDH1A1COMTKDM4E
SCHEMBL8186323 0.75 PPOX (0.38) CNR1L3MBTL1
SCHEMBL8192247 0.74 PPOX (0.36) ALDH1A1COMT
SCHEMBL8189134 0.73 TDP1 (0.35) HSD11B1ALDH1A1COMTKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6015774-A Pyrazin-2-one derivatives, their use, and intermediates for their production SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2000-01-18 US disclosed