SCHEMBL8192173

SCHEMBL8192173

O=C1N=CNC12CCNCC2c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.37
DRD2 P14416 1/20 0.37
SLC6A9 P48067 6/20 0.33
OPRM1 P35372 4/20 0.33
SLC6A5 Q9Y345 3/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
KDM1A O60341 4/20 0.33
MAOB P27338 3/20 0.33
MAOA P21397 1/20 0.32
NISCH Q9Y2I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037246 0.75 SIGMAR1 (0.40) SIGMAR1DRD2SLC6A9OPRM1SLC6A5
SCHEMBL2879213 0.74 SLC6A9 (0.38) SIGMAR1DRD2SLC6A9OPRM1SLC6A5
Hydrochloric Acid SCHEMBL9037991 0.73 SIGMAR1 (0.39) SIGMAR1DRD2SLC6A9OPRM1SLC6A5
SCHEMBL15568523 0.70 TAAR1 (0.41) SIGMAR1DRD2OPRM1MAPTTAAR1
SCHEMBL17135722 0.70 OPRM1 (0.44) SIGMAR1DRD2OPRM1MAPTTAAR1
SCHEMBL16221385 0.68 KDM1A (0.46) SIGMAR1DRD2OPRM1MAPTTAAR1
SCHEMBL32672366 0.68 KDM1A (0.41) SIGMAR1DRD2OPRM1MAPTTAAR1
SCHEMBL15571072 0.67 TAAR1 (0.39) SIGMAR1DRD2OPRM1MAPTTAAR1
Hydrochloric Acid SCHEMBL5505790 0.66 TAAR1 (0.39) DRD2MAPTTAAR1KDM1AMAOB
SCHEMBL1138335 0.64 SLC6A9 (0.56) SLC6A9OPRM1SLC6A5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO disclosed
EP-0696280-A1 SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES USEFUL AS TACHYKININ ANTAGONISTS MERRELL DOW PHARMA (US) 1996-02-14 EP disclosed
WO-1994026735-A1 SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES USEFUL AS TACHYKININ ANTAGONISTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-11-24 WO disclosed