SCHEMBL8195201

SCHEMBL8195201

CC1OC(=O)C(Oc2ccc(F)c(F)c2)=C1c1ccc(S(C)(=O)=O)c(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.44
PTGS1 P23219 1/20 0.44
PDE3B Q13370 11/20 0.40
PDE3A Q14432 11/20 0.40
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
ABCB11 O95342 1/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
KIF11 P52732 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
EPAS1 Q99814 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312284 0.83 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL6846585 0.73 PTGS2 (0.44) PTGS2PTGS1ALOX5APFEN1EPAS1
SCHEMBL6704623 0.69 PTGS2 (0.39) PTGS2PTGS1EPAS1
SCHEMBL6846488 0.66 PTGS2 (0.36) PTGS2PTGS1
SCHEMBL6739092 0.66 NR3C1 (0.52) PTGS2PTGS1
SCHEMBL6846588 0.65 PTGS2 (0.39) PTGS2PTGS1EPAS1
SCHEMBL6741612 0.63 PTGS2 (0.45) PTGS2PTGS1PDE3BPDE3A
SCHEMBL5208053 0.62 PTGS2 (0.80) PTGS2PTGS1
SCHEMBL5377415 0.62 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL5831189 0.62 KIF11 (0.44) PIK3CDPIK3CAPIK3CBPIK3CGABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6020343-A (Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitors MERCK FROSST CANADA, INC. (CA) 2000-02-01 US disclosed