SCHEMBL8196136

SCHEMBL8196136

CC(=O)OCS(=O)(=O)c1ccc(-c2[nH]nc(C(F)(F)F)c2-c2cccc(Cl)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.38
PLK4 O00444 2/20 0.38
RORC P51449 5/20 0.37
TRPV1 Q8NER1 1/20 0.36
FFAR1 O14842 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
IKBKE Q14164 1/20 0.33
DAPK3 O43293 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
EGFR P00533 1/20 0.33
RET P07949 1/20 0.33
PIM1 P11309 1/20 0.33
FER P16591 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33
MARK3 P27448 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8187466 0.85 PTGS2 (0.39) PTGS2SMN1; SMN2PTGS1
SCHEMBL8195827 0.84 PTGS2 (0.40) PTGS2MAPK1PTGS1
SCHEMBL8197121 0.83 PTGS2 (0.39) PTGS2PLK4RORCTRPV1IKBKE
SCHEMBL8200073 0.80 FFAR1 (0.35) PLK4TRPV1FFAR1CDK2AURKB
SCHEMBL8202072 0.80 PTGS2 (0.36) PTGS2PTGS1
SCHEMBL8200042 0.79 AR (0.37) RORCAURKB
SCHEMBL8201788 0.79 IDO1 (0.37) PTGS2PLK4RETCDK2PRKX
SCHEMBL8196138 0.77 PTGS2 (0.36) PTGS2TRPV1PTGS1
SCHEMBL8187580 0.77 TP53 (0.37) PTGS2SMN1; SMN2PTGS1PTGDR2
SCHEMBL8195825 0.76 PTGS2 (0.38) PTGS2SMN1; SMN2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed