SCHEMBL8196138

SCHEMBL8196138

CC(=O)OCS(=O)(=O)c1ccc(-c2[nH]nc(Cl)c2-c2ccc(F)c(C)c2)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.36
PTGS1 P23219 5/20 0.36
PHGDH O43175 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
MAPK14 Q16539 1/20 0.33
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202075 0.93 PTGS2 (0.37) PTGS2PTGS1MEN1HTTKMT2A
SCHEMBL8187580 0.87 TP53 (0.37) PTGS2PTGS1MEN1KMT2ATP53
SCHEMBL8200073 0.85 FFAR1 (0.35) TRPV1MAPK14MAPT
SCHEMBL8195877 0.84 PTGS2 (0.41) PTGS2PTGS1MAPK14
SCHEMBL8201788 0.82 IDO1 (0.37) PTGS2MEN1HTTKMT2ALMNA
SCHEMBL8188126 0.82 MEN1 (0.40) PTGS2PTGS1MEN1HTTKMT2A
SCHEMBL8196169 0.82 ALDH1A1 (0.37) PTGS2PTGS1PHGDHMEN1KMT2A
SCHEMBL8188503 0.82 PTGS2 (0.40) PTGS2PTGS1MAPK14
SCHEMBL8196136 0.77 PTGS2 (0.38) PTGS2PTGS1TRPV1
SCHEMBL8196142 0.76 PTGS2 (0.37) PTGS2PTGS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed