SCHEMBL8202072

SCHEMBL8202072

CC(=O)OCCS(=O)(=O)c1ccc(-c2[nH]nc(C(F)(F)F)c2-c2ccc(C)c(Cl)c2)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.36
PTGS1 P23219 4/20 0.36
NEK1 Q96PY6 1/20 0.34
CHUK O15111 1/20 0.33
CASP3 P42574 1/20 0.32
NOTUM Q6P988 1/20 0.32
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195825 0.89 PTGS2 (0.38) PTGS2PTGS1ALDH1A1HTT
SCHEMBL8194817 0.87 PTGS2 (0.40) PTGS2PTGS1CHUKALDH1A1CA2
SCHEMBL8228161 0.84 PPARD (0.35) PTGS2PTGS1CHUKNOTUMALDH1A1
SCHEMBL8195777 0.84 PTGS2 (0.37) PTGS2PTGS1ALDH1A1KDM4EHTT
SCHEMBL8187466 0.82 PTGS2 (0.39) PTGS2PTGS1ALDH1A1
SCHEMBL8196086 0.81 ALDH1A1 (0.39) NEK1ALDH1A1HPGDHTTCA2
SCHEMBL8200030 0.81 POLB (0.40) PTGS2PTGS1ALDH1A1KDM4EHPGD
SCHEMBL8196136 0.80 PTGS2 (0.38) PTGS2PTGS1
SCHEMBL8194813 0.78 PTGS2 (0.37) PTGS2ALDH1A1KDM4EHPGDHTT
SCHEMBL8196005 0.78 MEN1 (0.39) PTGS2PTGS1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed