SCHEMBL8201788

SCHEMBL8201788

CC(=O)OCS(=O)(=O)c1ccc(-c2[nH]nc(Cl)c2-c2cccc(Br)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.37
IKBKB O14920 1/20 0.34
DYRK1A Q13627 2/20 0.34
DYRK1B Q9Y463 2/20 0.34
PLK4 O00444 2/20 0.34
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34
MMP7 P09237 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
RET P07949 1/20 0.34
PRKX P51817 1/20 0.34
TAOK1 Q7L7X3 1/20 0.34
CDK2 P24941 1/20 0.33
MEN1 O00255 2/20 0.33
HPGD P15428 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200073 0.89 FFAR1 (0.35) PLK4CDK2MAPTALDH1A1L3MBTL1
SCHEMBL8187580 0.84 TP53 (0.37) MEN1KMT2AALDH1A1NEK1PTGS2
SCHEMBL8202075 0.83 PTGS2 (0.37) PLK4MEN1KMT2AMAPTHTT
SCHEMBL8196169 0.82 ALDH1A1 (0.37) MEN1KMT2AMAPTALDH1A1L3MBTL1
SCHEMBL8196138 0.82 PTGS2 (0.36) MEN1KMT2AMAPTLMNAHTT
SCHEMBL8188126 0.82 MEN1 (0.40) MEN1KMT2AALDH1A1HTTPTGS2
SCHEMBL8196136 0.79 PTGS2 (0.38) DYRK1APLK4RETPRKXCDK2
SCHEMBL8196005 0.73 MEN1 (0.39) MEN1KMT2AALDH1A1HTTPTGS2
SCHEMBL8195771 0.73 GRM5 (0.37) DYRK1ADYRK1BMEN1HPGDKMT2A
SCHEMBL8201297 0.72 L3MBTL1 (0.37) MEN1KMT2AMAPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed