SCHEMBL8196805

SCHEMBL8196805

Cc1ccc(S(=O)(=O)OC[C@H](O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.53
P2RX7 Q99572 2/20 0.47
PSEN1 P49768 3/20 0.46
PSEN2 P49810 3/20 0.46
APH1B Q8WW43 3/20 0.46
NCSTN Q92542 3/20 0.46
APH1A Q96BI3 3/20 0.46
PSENEN Q9NZ42 3/20 0.46
APP P05067 1/20 0.45
ATM Q13315 1/20 0.45
ALDH1A1 P00352 3/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 2/20 0.44
PKM P14618 2/20 0.44
HPGD P15428 2/20 0.44
HTT P42858 2/20 0.44
KMT2A Q03164 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
MEN1 O00255 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14189470 1.00 KLK5 (0.53) KLK5P2RX7PSEN1PSEN2APH1B
SCHEMBL8685847 1.00 KLK5 (0.53) KLK5P2RX7PSEN1PSEN2APH1B
SCHEMBL14209406 0.91 KLK5 (0.46) KLK5P2RX7PSEN1PSEN2APH1B
SCHEMBL3348635 0.87 ALDH1A1 (0.44) KLK5P2RX7ATMALDH1A1TSHR
SCHEMBL1258432 0.86 ATM (0.56) P2RX7APPATMALDH1A1TSHR
SCHEMBL1258429 0.86 ATM (0.56) P2RX7APPATMALDH1A1TSHR
SCHEMBL6562244 0.85 KLK5 (0.59) KLK5PSEN1PSEN2APH1BNCSTN
SCHEMBL6814107 0.85 KLK5 (0.59) KLK5PSEN1PSEN2APH1BNCSTN
SCHEMBL10209786 0.83 ALDH1A1 (0.46) KLK5P2RX7ATMALDH1A1TSHR
SCHEMBL7275804 0.80 CA2 (0.50) KLK5ATMALDH1A1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970066-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 2000-01-12 EP disclosed
WO-1998029401-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 1998-07-09 WO disclosed