SCHEMBL8196861

SCHEMBL8196861

COc1ccc(-c2c(Cl)n[nH]c2-c2ccc(S(=O)(=O)CCO)cc2)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.43
PTGS1 P23219 7/20 0.42
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AURKA O14965 1/20 0.38
NTRK1 P04629 1/20 0.38
KDR P35968 1/20 0.38
AURKB Q96GD4 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188096 0.94 PTGS2 (0.42) PTGS2PTGS1MEN1KMT2AAURKA
SCHEMBL8196687 0.90 PTGS2 (0.41) PTGS2PTGS1ALDH1A1LMNARAB9A
SCHEMBL8196703 0.88 PTGS2 (0.42) PTGS2PTGS1KMT2AALDH1A1LMNA
SCHEMBL8196005 0.87 MEN1 (0.39) PTGS2PTGS1MEN1KMT2AAURKA
SCHEMBL8199737 0.86 PTGS2 (0.40) PTGS2PTGS1ALDH1A1LMNA
SCHEMBL8196014 0.86 ALDH1A1 (0.37) PTGS2AURKANTRK1KDRAURKB
SCHEMBL8188126 0.85 MEN1 (0.40) PTGS2PTGS1MEN1KMT2AAURKA
SCHEMBL8058037 0.85 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL8197292 0.84 PTGS2 (0.40) PTGS2PTGS1ALDH1A1
SCHEMBL8194835 0.82 PTGS2 (0.41) PTGS2PTGS1ALDH1A1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed