SCHEMBL8196014

SCHEMBL8196014

COc1cc(-c2c(Cl)n[nH]c2-c2ccc(S(=O)(=O)CCCO)cc2)ccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
AURKA O14965 1/20 0.36
NTRK1 P04629 1/20 0.36
KDR P35968 1/20 0.36
AURKB Q96GD4 1/20 0.36
CA2 P00918 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
PKM P14618 2/20 0.35
SCN9A Q15858 1/20 0.35
FYN P06241 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
PHGDH O43175 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGS2 P35354 1/20 0.34
TSHR P16473 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
KMO O15229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188096 0.92 PTGS2 (0.42) AURKANTRK1KDRAURKBPTGDR2
SCHEMBL8196899 0.87 PTGS2 (0.39) ALDH1A1CA2PTGDR2PTGS2
SCHEMBL8196861 0.86 PTGS2 (0.43) ALDH1A1AURKANTRK1KDRAURKB
SCHEMBL8200031 0.85 PTGS2 (0.39) ALDH1A1MAPTCA2PTGDR2PTGS2
SCHEMBL8196169 0.83 ALDH1A1 (0.37) ALDH1A1MAPTAURKANTRK1KDR
SCHEMBL8196062 0.82 ALDH1A1 (0.46) ALDH1A1MAPTCA2SMN1; SMN2PTGS2
SCHEMBL8196010 0.82 CA2 (0.43) CA2PTGDR2PTGS2
SCHEMBL8187634 0.82 GRM5 (0.38) ALDH1A1MAPTAURKANTRK1KDR
SCHEMBL8196195 0.81 PTGS2 (0.40) AURKBCA2FYNPTGDR2MAPK1
SCHEMBL8194835 0.81 PTGS2 (0.41) ALDH1A1SMN1; SMN2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed